Lestaurtinib

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Lestaurtinib
Systematic (IUPAC) name
?
Identifiers
CAS number	?
ATC code	?
PubChem	126565
Chemical data
Formula	C26H21N3O4
Mol. mass	439.462 g/mol
Pharmacokinetic data
Bioavailability	?
Metabolism	?
Half life	?
Excretion	?
Therapeutic considerations
Pregnancy cat.	?
Legal status
Routes	?

Lestaurtinib (rINN, codenamed CEP-701) is a tyrosine kinase inhibitor undergoing research for the treatment of acute myelogenous leukemia (AML) and myeloproliferative disorders. It is an analog of staurosporine.

As of 2008, it is currently in Phase III clinical trials for AML and Phase II clinical trials for myeloproliferative disorders. ^[1]

It is being developed by Cephalon.

[edit] References

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