Talk:Lapatinib

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[edit] The

"The exact site of binding has currently not been confirmed (EGFR and ErbB2 have a number of intracellular phosphorylation sites)."

-- this should probably be removed, at least for EGFR, since there's a crystal structure of Lapatinib bound to the ATP binding site from 2004: pdb code 1XKK.

Lapatinib is well known as an ATP-competitive kinase inhibitor (that was determined well before the crystal structure being solved). The comment has been removed. 05:52, 18 December 2007 (UTC)btavshan

Its identity as a kinase inhibitor is explicated in the third paragraph, if that wasn't obvious enough from the name. Could you point to when/where/what was actually removed? Otherwise, I can't tell if any information is missing that could go in there. Someguy1221 (talk) 05:57, 18 December 2007 (UTC)